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threo Ifenprodil hemitartrate, Tocris Bioscience™

NR2B-selective NMDA antagonist; also σ agonist

Marke:  Tocris (Bio-Techne) 289250

Weitere Details : Netto-Gewicht : 0.01000kg

Menge. 50mg

 Weitere Artikel aus diesem Sortiment

Artikelnummer. 13411994

  • 857.56 € / 50 Milligramm


Voraussichtlicher Liefertermin 27-06-2019
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Beschreibung

Beschreibung

Potent σ receptor agonist (K i values are 59.1 and 2 nM for σ1 and σ2 receptors respectively) and GluN2B (formally NR2B) subunit-selective NMDA receptor antagonist (IC 50 values are 0.22 and 324.8 μM at GluN2B and GluN2A respectively). Displays ∽8-fold reduced affinity at α-adrenoceptors compared to Ifenprodil (Cat.No. 0545). Inhibits the hERG potassium channel (IC 50 = 88 nM) and exhibits antiarrhythmic activity in vivo. Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.
Spezifikation

Chemische Identifikatoren

1312991-83-5
1601.98
threo ifenprodil hemitartrate
4-[(1S,2S)-2-(4-benzylpiperidin-1-yl)-1-hydroxypropyl]phenol;4-[(1R,2R)-2-(4-benzylpiperidin-1-yl)-1-hydroxypropyl]phenol;2,3-dihydroxybutanedioic acid
C92H120N4O20
MMUFFGLAKFWLGJ-RRQZTXAJSA-N
90488783
CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.C(C(C(=O)O)O)(C(=O)O)O.C(C(C(=O)O)O)(C(=O)O)O

Spezifikation

threo Ifenprodil hemitartrate
1312991-83-5
threo ifenprodil hemitartrate
CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.CC(C(C1=CC=C(C=C1)O)O)N2CCC(CC2)CC3=CC=CC=C3.C(C(C(=O)O)O)(C(=O)O)O.C(C(C(=O)O)O)(C(=O)O)O
1601.98
400.49
50mg
C92H120N4O20
MMUFFGLAKFWLGJ-RRQZTXAJSA-N
4-[(1S,2S)-2-(4-benzylpiperidin-1-yl)-1-hydroxypropyl]phenol;4-[(1R,2R)-2-(4-benzylpiperidin-1-yl)-1-hydroxypropyl]phenol;2,3-dihydroxybutanedioic acid
90488783
>98%
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