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Tocris Bioscience™ MOMBA

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Menge:
250 mg
Packungsgröße:
250 Milligramm
Beskrivning
MOMBA is a selective orthosteric agonist for human free fatty acid 2 (hFFA2) engineered receptors, designer receptors activated by designer drugs (DREADD), it shows no activity to wild-type hFFA2, hFFA3, and mouse FFA2. MOMBA inhibit forskolin-stimulated cAMP levels in cells expressing the hFFA2-DREADD receptor with improved potency and equivalent efficacy to Sorbic acid (Cat. No. 7119). In hFFA2-DREADD transgenic mice, MOMBA treatment significantly reduces gut transit and promotes concentration-dependent release of GLP-1 from colonic crypts. Orally bioavailable.
Specifikationer
Specifikationer
| Chemischer Name oder Material | 4-Methoxy-3-methylbenzoic acid |
| CAS | 6880-04-2 |
| Menge | 250 mg |
| Ziel | DREADD Activators |
| Summenformel | C9H10O3 |
| Reinheit | 0.98 |
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