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Tocris Bioscience™ Clobenpropit dihydrobromide
Highly potent H3 antagonist and H4 partial agonist
N.V.
Spezifikation
Prozentgehaltsbereich | >99% |
---|---|
Chemischer Name oder Material | N-(4-Chlorobenzyl)-S-[3-(4(5)-imidazolyl)propyl]isothiourea dihydrobromide |
CAS | 145231-35-2 |
Beschreibung
An extremely potent histamine H3 antagonist/inverse agonist (pA2=9.93). Also displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM.Spezifikation
>99% | |
N-(4-Chlorobenzyl)-S-[3-(4(5)-imidazolyl)propyl]isothiourea dihydrobromide | |
145231-35-2 |
For Research Use Only